Items where Author is "Gmeiner, Peter"

Article

Lahmy, Ranit and Huebner, Harald and Gmeiner, Peter and Koenig, Burkhard (2024) Covalent and Visible-Light Photoswitchable Derivatives of the Potent Synthetic Opioid Isotonitazene and Other Nitazenes. CHEMPHOTOCHEM, 8 (7). e202400022. ISSN 2367-0932,

Ertl, Fabian J. and Kopanchuk, Sergei and Dijon, Nicola C. and Veiksina, Santa and Tahk, Maris-Johanna and Laasfeld, Tonis and Schettler, Franziska and Gattor, Albert O. and Huebner, Harald and Archipowa, Nataliya and Koeckenberger, Johannes and Heinrich, Markus R. and Gmeiner, Peter and Kutta, Roger J. and Holliday, Nicholas D. and Rinken, Ago and Keller, Max (2024) Dually Labeled Neurotensin NTS1R Ligands for Probing Radiochemical and Fluorescence-Based Binding Assays. JOURNAL OF MEDICINAL CHEMISTRY, 67 (18). pp. 16664-16691. ISSN 0022-2623, 1520-4804

Lahmy, Ranit and Hübner, Harald and Schmidt, Maximilian F. and Lachmann, Daniel and Gmeiner, Peter and König, Burkhard (2022) Photochromic Fentanyl Derivatives for Controlled mu-Opioid Receptor Activation. CHEMISTRY-A EUROPEAN JOURNAL, 28 (63): e202201515. ISSN 0947-6539, 1521-3765

Tropmann, Katharina and Bresinsky, Merlin and Forster, Lisa and Moennich, Denise and Buschauer, Armin and Wittmann, Hans-Joachim and Huebner, Harald and Gmeiner, Peter and Pockes, Steffen and Strasser, Andrea (2021) Abolishing Dopamine D-2long/D-3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H-2 Receptor Agonists. JOURNAL OF MEDICINAL CHEMISTRY, 64 (12). pp. 8684-8709. ISSN 0022-2623, 1520-4804

Weinhart, Corinna G. and Wifling, David and Schmidt, Maximilian F. and Neu, Eduard and Hoering, Carina and Clark, Timothy and Gmeiner, Peter and Keller, Max (2021) Dibenzodiazepinone-type muscarinic receptor antagonists conjugated to basic peptides: Impact of the linker moiety and unnatural amino acids on M2R selectivity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 213: 113159. ISSN 0223-5234, 1768-3254

Konieczny, Adam and Conrad, Marcus and Ertl, Fabian J. and Gleixner, Jakob and Gattor, Albert O. and Graetz, Lukas and Schmidt, Maximilian F. and Neu, Eduard and Horn, Anselm H. C. and Wifling, David and Gmeiner, Peter and Clark, Timothy and Sticht, Heinrich and Keller, Max (2021) N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y-4 Receptor Ligands Results in Picomolar Binding Constants. JOURNAL OF MEDICINAL CHEMISTRY, 64 (22). pp. 16746-16769. ISSN 0022-2623, 1520-4804

Keller, Max and Mahuroof, Shahani A. and Yee, Vivyanne Hong and Carpenter, Jessica and Schindler, Lisa and Littmann, Timo and Pegoli, Andrea and Huebner, Harald and Bernhardt, Guenther and Gmeiner, Peter and Holliday, Nicholas D. (2020) Fluorescence Labeling of Neurotensin(8-13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity. ACS MEDICINAL CHEMISTRY LETTERS, 11 (1). pp. 16-22. ISSN 1948-5875

She, Xueke and Pegoli, Andrea and Gruber, Corinna G. and Wifling, David and Carpenter, Jessica and Huebner, Harald and Chen, Mengya and Wan, Jianfei and Bernhardt, Guenther and Gmeiner, Peter and Holliday, Nicholas D. and Keller, Max (2020) Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M-2 Receptor. JOURNAL OF MEDICINAL CHEMISTRY, 63 (8). pp. 4133-4154. ISSN 0022-2623, 1520-4804

Stolwijk, Judith A. and Mildner, Anne-Kathrin and Kade, Christian and Skiba, Michael and Bernhardt, Guenther and Buschauer, Armin and Huebner, Harald and Gmeiner, Peter and Wegener, Joachim (2020) Stepwise Dosing Protocol for Increased Throughput in Label-Free Impedance-Based GPCR Assays. JOVE-JOURNAL OF VISUALIZED EXPERIMENTS (156): e60686. ISSN 1940-087X

Gienger, Marie and Huebner, Harald and Loeber, Stefan and Koenig, Burkhard and Gmeiner, Peter (2020) Structure-based development of caged dopamine D-2/D-3 receptor antagonists. SCIENTIFIC REPORTS, 10 (1). ISSN 2045-2322

Pegoli, Andrea and Wifling, David and Gruber, Corinna G. and She, Xueke and Huebner, Harald and Bernhardt, Guenther and Gmeiner, Peter and Keller, Max (2019) Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity. JOURNAL OF MEDICINAL CHEMISTRY, 62 (11). pp. 5358-5369. ISSN 0022-2623, 1520-4804

She, Xueke and Pegoli, Andrea and Mayr, Judith and Huebner, Harald and Bernhardt, Guenther and Gmeiner, Peter and Keller, Max (2017) Heterodimerization of Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Leads to Increased M2R Affinity and Selectivity. ACS OMEGA, 2 (10). pp. 6741-6754. ISSN 2470-1343

Simeth, Nadja A. and Bause, Manuel and Dobmeier, Michael and Kling, Ralf C. and Lachmann, Daniel and Huebner, Harald and Einsiedel, Juergen and Gmeiner, Peter and Koenig, Burkhard (2017) NTS2-selective neurotensin mimetics with tetrahydrofuran amino acids. BIOORGANIC & MEDICINAL CHEMISTRY, 25 (1). pp. 350-359. ISSN 0968-0896, 1464-3391

Lachmann, Daniel and Studte, Carolin and Maennel, Barbara and Huebner, Harald and Gmeiner, Peter and Koenig, Burkhard (2017) Photochromic Dopamine Receptor Ligands Based on Dithienylethenes and Fulgides. CHEMISTRY-A EUROPEAN JOURNAL, 23 (54). pp. 13423-13434. ISSN 0947-6539, 1521-3765

Pegoli, Andrea and She, Xueke and Wifling, David and Huebner, Harald and Bernhardt, Guenther and Gmeiner, Peter and Keller, Max (2017) Radiolabeled Dibenzodiazepinone-Type Antagonists Give Evidence of Dualsteric Binding at the M-2 Muscarinic Acetylcholine Receptor. JOURNAL OF MEDICINAL CHEMISTRY, 60 (8). pp. 3314-3334. ISSN 0022-2623, 1520-4804

Naporra, Franziska and Gobleder, Susanne and Wittmann, Hans Joachim and Spindler, Julia and Bodensteiner, Michael and Bernhardt, Guenther and Huebner, Harald and Gmeiner, Peter and Elz, Sigurd and Strasser, Andrea (2016) Dibenzo[bf][1,4]oxazepines and dibenzo[b,e]oxepines: Influence of the chlorine substitution pattern on the pharmacology at the H1R, H4R, 5-HT2AR and other selected GPCRs. PHARMACOLOGICAL RESEARCH, 113. pp. 610-625. ISSN 1043-6618

Keller, Max and Kuhn, Kilian K. and Einsiedel, Juergen and Huebner, Harald and Biselli, Sabrina and Mollereau, Catherine and Wifling, David and Svobodova, Jaroslava and Bernhardt, Guenther and Cabrele, Chiara and Vanderheyden, Patrick M. L. and Gmeiner, Peter and Buschauer, Armin (2016) Mimicking of Arginine by Functionalized N-omega-Carbamoylated Arginine As a New Broadly Applicable Approach to Labeled Bioactive Peptides: High Affinity Angiotensin, Neuropeptide Y, Neuropeptide FF, and Neurotensin Receptor Ligands As Examples. JOURNAL OF MEDICINAL CHEMISTRY, 59 (5). pp. 1925-1945. ISSN 0022-2623, 1520-4804

Loeber, Stefan and Huebner, Harald and Buschauer, Armin and Sanna, Fabrizio and Argiolas, Antonio and Melis, Maria Rosaria and Gmeiner, Peter (2012) Novel azulene derivatives for the treatment of erectile dysfunction. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 22 (23). pp. 7151-7154. ISSN 0960-894X