Items where Author is "Littmann, Timo"

Article

Tropmann, Katharina and Seibel-Ehlert, Ulla and Littmann, Timo and Strasser, Andrea (2021) Shining light on the histamine H-2 receptor: Synthesis of carbamoylguanidine-type agonists as a pharmacological tool to study internalization. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 52: 128388. ISSN 0960-894X, 1464-3405

Keller, Max and Mahuroof, Shahani A. and Yee, Vivyanne Hong and Carpenter, Jessica and Schindler, Lisa and Littmann, Timo and Pegoli, Andrea and Huebner, Harald and Bernhardt, Guenther and Gmeiner, Peter and Holliday, Nicholas D. (2020) Fluorescence Labeling of Neurotensin(8-13) via Arginine Residues Gives Molecular Tools with High Receptor Affinity. ACS MEDICINAL CHEMISTRY LETTERS, 11 (1). pp. 16-22. ISSN 1948-5875

Biselli, Sabrina and Alencastre, Ines and Tropmann, Katharina and Erdmann, Daniela and Chen, Mengya and Littmann, Timo and Maia, Andre F. and Gomez-Lazaro, Maria and Tanaka, Miho and Ozawa, Takeaki and Keller, Max and Lamghari, Meriem and Buschauer, Armin and Bernhardt, Guenther (2020) Fluorescent H-2 Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications. ACS MEDICINAL CHEMISTRY LETTERS, 11 (8). pp. 1521-1528. ISSN 1948-5875

Bartole, Edith and Graetz, Lukas and Littmann, Timo and Wifling, David and Seibel, Ulla and Buschauer, Armin and Bernhardt, Guenther (2020) UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H-3 and H-4 Receptors. JOURNAL OF MEDICINAL CHEMISTRY, 63 (10). pp. 5297-5311. ISSN 0022-2623, 1520-4804

Agnetta, Luca and Bermudez, Marcel and Riefolo, Fabio and Matera, Carlo and Claro, Enrique and Messerer, Regina and Littmann, Timo and Wolber, Gerhard and Holzgrabe, Ulrike and Decker, Michael (2019) Fluorination of Photoswitchable Muscarinic Agonists Tunes Receptor Pharmacology and Photochromic Properties. JOURNAL OF MEDICINAL CHEMISTRY, 62 (6). pp. 3009-3020. ISSN 0022-2623, 1520-4804

Bartole, Edith and Littmann, Timo and Tanaka, Miho and Ozawa, Takeaki and Buschauer, Armin and Bernhardt, Guenther (2019) [H-3]UR-DEBa176: A 2,4-Diaminopyrimidine-Type Radioligand Enabling Binding Studies at the Human, Mouse, and Rat Histamine H-4 Receptors. JOURNAL OF MEDICINAL CHEMISTRY, 62 (17). pp. 8338-8356. ISSN 0022-2623, 1520-4804

Schramm, Simon and Agnetta, Luca and Bermudez, Marcel and Gerwe, Hubert and Irmen, Matthias and Holze, Janine and Littmann, Timo and Wolber, Gerhard and Traenkle, Christian and Decker, Michael (2019) Novel BQCA- and TBPB-Derived M-1 Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism. CHEMMEDCHEM, 14 (14). pp. 1349-1358. ISSN 1860-7179, 1860-7187

Littmann, Timo and Buschauer, Armin and Bernhardt, Gunther (2019) Split luciferase-based assay for simultaneous analyses of the ligand concentration- and time-dependent recruitment of beta-arrestin2. ANALYTICAL BIOCHEMISTRY, 573. pp. 8-16. ISSN 0003-2697, 1096-0309

Schramm, Andrea and Mueller-Thuemen, Philip and Littmann, Timo and Harloff, Manuela and Ozawa, Takeaki and Schlossmann, Jens (2018) Establishing a Split Luciferase Assay for Proteinkinase G (PKG) Interaction Studies. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 19 (4): 1180. ISSN 1422-0067

Yang, Zhenlin and Han, Shuo and Keller, Max and Kaiser, Anette and Bender, Brian J. and Bosse, Mathias and Burkert, Kerstin and Koegler, Lisa M. and Wifling, David and Bernhardt, Guenther and Plank, Nicole and Littmann, Timo and Schmidt, Peter and Yi, Cuiying and Li, Beibei and Ye, Sheng and Zhang, Rongguang and Xu, Bo and Larhammar, Dan and Stevens, Raymond C. and Huster, Daniel and Meiler, Jens and Zhao, Qiang and Beck-Sickinger, Annette G. and Buschauer, Armin and Wu, Beili (2018) Structural basis of ligand binding modes at the neuropeptide Y Y-1 receptor. NATURE, 556 (7702). 520-+. ISSN 0028-0836, 1476-4687

Littmann, Timo and Ozawa, Takeaki and Hoffmann, Carsten and Buschauer, Armin and Bernhardt, Guenther (2018) A split luciferase-based probe for quantitative proximal determination of G alpha(q) signalling in live cells. SCIENTIFIC REPORTS, 8: 17179. ISSN 2045-2322

Dukorn, Stefanie and Littmann, Timo and Keller, Max and Kuhn, Kilian and Cabrele, Chiara and Baumeister, Paul and Bernhardt, Guenther and Buschauer, Armin (2017) Fluorescence- and Radiolabeling of [Lys(4),Nle(17,30)]hPP Yields Molecular Tools for the NPY Y-4 Receptor. BIOCONJUGATE CHEMISTRY, 28 (4). pp. 1291-1304. ISSN 1043-1802

Kuhn, Kilian K. and Littmann, Timo and Dukorn, Stefanie and Tanaka, Miho and Keller, Max and Ozawa, Takeaki and Bernhardt, Gunther and Buschauer, Armin (2017) In Search of NPY Y4R Antagonists: Incorporation of Carbamoylated Arginine, Aza-Amino Acids, or D-Amino Acids into Oligopeptides Derived from the C-Termini of the Endogenous Agonists. ACS OMEGA, 2 (7). pp. 3616-3631. ISSN 2470-1343

Reinartz, Michael T. and Kaelble, Solveig and Littmann, Timo and Ozawa, Takeaki and Dove, Stefan and Kaever, Volkhard and Wainer, Irving W. and Seifert, Roland (2015) Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the beta(2)-adrenoceptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 388 (1). pp. 51-65. ISSN 0028-1298, 1432-1912

Conference or Workshop Item

Hoering, Carina and Seibel, Ulla and Littmann, Timo and Graetz, Lukas and Strasser, Andrea and Bernhardt, Guenther (2020) A MiniG Protein Recruitment Assay for the Histamine Receptor Family to Functionally Characterize Histamine Receptor Ligands. In: Annual Meeting on Experimental Biology, APR 04-07, 2020, San Diego, CA.

Other

Reinartz, Michael T. and Littmann, Timo and Wainer, Irving William and Ozawa, Takeaki and Dove, Stefan and Seifert, Roland (2014) Quantifying ligand bias of enantiopure fenoterol derivatives in molecular and cellular beta(2)-adrenergic assay systems. SPRINGER, NEW YORK.