Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry I (Prof. Elz)" and Year is 2002

B

Beckers, Thomas and Reissmann, Thomas and Schmidt, Mathias and Burger, Angelika M. and Fiebig, Heinz H. and Vanhoefer, Udo and Pongratz, Herwig and Hufsky, Harald and Hockemeyer, Jörg and Frieser, Markus and Mahboobi, Siavosh (2002) 2-aroylindoles, a novel class of potent, orally active small molecule tubulin inhibitors. CANCER RESEARCH, 62 (11). pp. 3113-3119. ISSN 0008-5472, 1538-7445

E

El-Subbagh, Hussein and Wittig, Thomas and Decker, Michael and Elz, Sigurd and Nieger, Martin and Lehmann, Jochen (2002) Dopamine/serotonin receptor ligands. Part IV [1]: Synthesis and pharmacology of novel 3-benzazecines and 3-benzazonines as potential 5-HT2A and dopamine receptor ligands. ARCHIV DER PHARMAZIE, 335 (9). pp. 443-448. ISSN 0365-6233, 1521-4184

Elz, S. and Klaess, T. and Heim, R. and Warnke, U. and Pertz, H. H. (2002) Development of highly potent partial agonists and chiral antagonists as tools for the study of 5-HT2A-receptor mediated functions. In: 43rd Spring Meeting Deutsche Gesellschaft für experimentelle und klinische Pharmakologie und Toxikologie, March 12-14, 2002, Mainz.

G

Grassmann, Sven and Sadek, Bassem and Ligneau, Xavier and Elz, Sigurd and Ganellin, C. Robin and Arrang, Jean-Michel and Schwartz, Jean-Charles and Stark, Holger and Schunack, Walter (2002) Progress in the proxifan class: heterocyclic congeners as novel potent and selective histamine H-3-receptor antagonists. EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 15 (4): PII S0928-. pp. 367-378. ISSN 0928-0987, 1879-0720

L

Lazewska, Dorota and Kiec-Kononowicz, Katarzyna and Pertz, H. H. and Elz, Sigurd and Stark, Holger and Schunack, W. (2002) Piperidine-containing histamine H-3 receptor antagonists of the carbamate series: the influence of the additional ether functionality. PHARMAZIE, 57 (12). pp. 791-795. ISSN 0031-7144

Letzel, Matthias C. and Gruetzmacher, Hans-Friedrich and Fuerst, Thomas and Mayer, Klaus K. and Wiegrebe, Wolfgang (2002) Functional group migration in benzaldoxime-O-n-propyl ether radical cation. INTERNATIONAL JOURNAL OF MASS SPECTROMETRY, 217 (1-3): PII S1387-. pp. 153-168. ISSN 1387-3806

M

Mahboobi, Siavosh and Teller, Steffen and Pongratz, Herwig and Hufsky, Harald and Sellmer, Andreas and Botzki, Alexander and Uecker, Andrea and Beckers, Thomas and Baasner, Silke and Schaechtele, Christoph and Ueberall, Florian and Kassack, Matthias U. and Dove, Stefan and Boehmer, Frank-D. (2002) Bis(1H-2-indolyl)methanones as a novel class of inhibitors of the platelet-derived growth factor receptor kinase. JOURNAL OF MEDICINAL CHEMISTRY, 45 (5). pp. 1002-1018. ISSN 0022-2623, 1520-4804

Menghin, S. and Kramer, K. and Pertz, H. H. and Schunack, W. and Elz, S. (2002) Arylalkyl and heteroarylalkyl analogues of suprahistaprodifen are potent histamine H-1-receptor agonists in vitro. In: 43rd Spring Meeting Deutsche Gesellschaft für experimentelle und klinische Pharmakologie und Toxikologie, March 12-14, 2002, Mainz.

S

Sasse, Astrid and Ligneau, Xavier and Rouleau, Agnes and Elz, Sigurd and Ganellin, C. Robin and Arrang, Jean-Michel and Schwartz, Jean-Charles and Schunack, Walter and Stark, Holger (2002) Influence of bulky substituents on histamine H-3 receptor agonist/antagonist properties. JOURNAL OF MEDICINAL CHEMISTRY, 45 (18): UNSP JM020. pp. 4000-4010. ISSN 0022-2623

Seifert, R. and Buerckstuemmer, T. and Buschauer, A. and Pertz, H. H. and Schunack, W. and Elz, S. (2002) Multiple pharmacological differences between the human and guinea pig histamine H-1-receptor. In: 43rd Spring Meeting Deutsche Gesellschaft für experimentelle und klinische Pharmakologie und Toxikologie, March 12-14, 2002, Mainz.

T

Teller, S. and Kraemer, D. and Boehmer, S. A. and Tse, K. F. and Small, D. and Mahboobi, Siavosh and Wallrapp, C. and Beckers, T. and Kratz-Albers, K. and Schwable, J. and Serve, H. and Boehmer, F. D. (2002) Bis(1 H-2-indolyl)-1-methanones as inhibitors of the hematopoietic tyrosine kinase Flt3. LEUKEMIA, 16 (8). pp. 1528-1534. ISSN 0887-6924