Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry I (Prof. Elz)" and Year is 2010

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Birnkammer, T. and Kraus, A. and Preuss, H. and Bernhardt, G. and Dove, S. and Elz, S. and Seifert, R. and Buschauer, A. (2010) APPLICATION OF THE BIVALENT LIGAND APPROACH TO ACYLGUANIDINES RESULTED IN HIGHLY POTENT AND SELECTIVE HISTAMINE H-2 RECEPTOR AGONISTS. INFLAMMATION RESEARCH, 59 (4Suppl). S353. ISSN 1023-3830

Brunskole, I. and Strasser, A. and Buschauer, A. and Seifert, R. (2010) Contribution of extracellular domains to ligand-receptor interactions at the human histamine H-4-receptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 381 (1Suppl). p. 13. ISSN 0028-1298

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Ghorai, Prasanta and Kraus, Anja and Birnkammer, Tobias and Geyer, Roland and Bernhardt, Guenther and Dove, Stefan and Seifert, Roland and Elz, Sigurd and Buschauer, Armin (2010) Chiral N-G-acylated hetarylpropylguanidine-type histamine H-2 receptor agonists do not show significant stereoselectivity. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 20 (10). pp. 3173-3176. ISSN 0960-894X

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Jandt, Enrico and Mutschke, Oliver and Mahboobi, Siavosh and Uecker, Andrea and Platz, Ronny and Berndt, Alexander and Boehmer, Frank-D. and Figulla, Hans R. and Werner, Gerald S. (2010) Stent-based release of a selective PDGF-receptor blocker from the bis-indolylmethanon class inhibits restenosis in the rabbit animal model. VASCULAR PHARMACOLOGY, 52 (1-2). pp. 55-62. ISSN 1537-1891

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Mahboobi, Siavosh and Sellmer, Andreas and Winkler, Matthias and Eichhorn, Emerich and Pongratz, Herwig and Ciossek, Thomas and Baer, Thomas and Maier, Thomas and Beckers, Thomas (2010) Novel Chimeric Histone Deacetylase Inhibitors: A Series of Lapatinib Hybrides as Potent Inhibitors of Epidermal Growth Factor Receptor (EGFR), Human Epidermal Growth Factor Receptor 2 (HER2), and Histone Deacetylase Activity. JOURNAL OF MEDICINAL CHEMISTRY, 53 (24). pp. 8546-8555. ISSN 0022-2623

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Schneider, Erich H. and Schnell, David and Strasser, Andrea and Dove, Stefan and Seifert, Roland (2010) Impact of the DRY Motif and the Missing "Ionic Lock" on Constitutive Activity and G-Protein Coupling of the Human Histamine H-4 Receptor. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 333 (2). pp. 382-392. ISSN 0022-3565

Schneider, Erich H. and Strasser, Andrea and Thurmond, Robin L. and Seifert, Roland (2010) Structural Requirements for Inverse Agonism and Neutral Antagonism of Indole-, Benzimidazole-, and Thienopyrrole-Derived Histamine H-4 Receptor Ligands. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 334 (2). pp. 513-521. ISSN 0022-3565, 1521-0103

Strasser, Andrea and Wittmann, Hans-Joachim (2010) 3D-QSAR CoMFA Study to Predict Orientation of Suprahistaprodifens and Phenoprodifens in the Binding-Pocket of Four Histamine H-1-Receptor Species. MOLECULAR INFORMATICS, 29 (4). pp. 333-341. ISSN 1868-1743

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Uecker, Andrea and Sicker, Marit and Beckers, Thomas and Mahboobi, Siavosh and Hagerstrand, Daniel and Ostman, Arne and Boehmer, Frank-D. (2010) Chimeric tyrosine kinase-HDAC inhibitors as antiproliferative agents. ANTI-CANCER DRUGS, 21 (8). pp. 759-765. ISSN 0959-4973