Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer)" and Year is 2011

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Birnkammer, T. and Kraus, A. and Bernhardt, G. and Dove, S. and Elz, S. and Seifert, R. and Buschauer, A. (2011) SYNTHESIS AND STRUCTURE ACTIVITY RELATIONSHIPS OF BIVALENT ACYLGUANIDINE-TYPE HISTAMINE H-2 RECEPTOR AGONISTS. INFLAMMATION RESEARCH, 60 (Suppl2). S354-S355. ISSN 1023-3830

Braun, Stephan and Botzki, Alexander and Salmen, Sunnhild and Textor, Christian and Bernhardt, Guenther and Dove, Stefan and Buschauer, Armin (2011) Design of benzimidazole- and benzoxazole-2-thione derivatives as inhibitors of bacterial hyaluronan lyase. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 46 (9). pp. 4419-4429. ISSN 0223-5234

Brunskole, I. and Strasser, A. and Seifert, R. and Buschauer, A. (2011) SECOND AND THIRD EXTRACELLULAR LOOPS OF THE HISTAMINE H-4 RECEPTOR ARE INVOLVED IN RECEPTOR ACTIVATION. INFLAMMATION RESEARCH, 60 (Suppl2). S354. ISSN 1023-3830

Brunskole, Irena and Strasser, Andrea and Seifert, Roland and Buschauer, Armin (2011) Role of the second and third extracellular loops of the histamine H-4 receptor in receptor activation. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 384 (3). pp. 301-317. ISSN 0028-1298

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Ferstl, Matthias and Strasser, Andrea and Wittmann, Hans-Joachim and Drechsler, Markus and Rischer, Matthias and Engel, Juergen and Goepferich, Achim (2011) Nanofibers Resulting from Cooperative Electrostatic and Hydrophobic Interactions between Peptides and Polyelectrolytes of Opposite Charge. LANGMUIR, 27 (23). pp. 14450-14459. ISSN 0743-7463

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Geduhn, Jens and Dove, Stefan and Shen, Yuequan and Tang, Wei-Jen and Koenig, Burkhard and Seifert, Roland (2011) Bis-Halogen-Anthraniloyl-Substituted Nucleoside 5 '-Triphosphates as Potent and Selective Inhibitors of Bordetella pertussis Adenylyl Cyclase Toxin. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 336 (1). pp. 104-115. ISSN 0022-3565, 1521-0103

Geyer, R. and Igel, P. and Buschauer, A. (2011) BIOISOSTERIC REPLACEMENT OF IMIDAZOLE IN CYANOGUANIDINE-TYPE hH(4)R AGONISTS-AN APPROACH TO IMPROVE H4R SELECTIVITY. INFLAMMATION RESEARCH, 60 (Suppl2). S353-S354. ISSN 1023-3830

Geyer, Roland and Buschauer, Armin (2011) Synthesis and Histamine H3 and H4 Receptor Activity of Conformationally Restricted Cyanoguanidines Related to UR-PI376. ARCHIV DER PHARMAZIE, 344 (12). pp. 775-785. ISSN 0365-6233, 1521-4184

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Keller, Max and Bernhardt, Guenther and Buschauer, Armin (2011) [H-3]UR-MK136: A Highly Potent and Selective Radioligand for Neuropeptide Y Y-1 Receptors. CHEMMEDCHEM, 6 (9). pp. 1566-1571. ISSN 1860-7179, 1860-7187

Keller, Max and Erdmann, Daniela and Pop, Nathalie and Pluym, Nikola and Teng, Shangjun and Bernhardt, Guenther and Buschauer, Armin (2011) Red-fluorescent argininamide-type NPY Y-1 receptor antagonists as pharmacological tools. BIOORGANIC & MEDICINAL CHEMISTRY, 19 (9). pp. 2859-2878. ISSN 0968-0896, 1464-3391

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Pluym, Nikola and Brennauer, Albert and Keller, Max and Ziemek, Ralf and Pop, Nathalie and Bernhardt, Guenther and Buschauer, Armin (2011) Application of the Guanidine-Acylguanidine Bioisosteric Approach to Argininamide-Type NPY Y-2 Receptor Antagonists. CHEMMEDCHEM, 6 (9). pp. 1727-1738. ISSN 1860-7179

Pop, Nathalie and Igel, Patrick and Brennauer, Albert and Cabrele, Chiara and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin (2011) Functional reconstitution of human neuropeptide Y (NPY) Y-2 and Y-4 receptors in Sf9 insect cells. JOURNAL OF RECEPTORS AND SIGNAL TRANSDUCTION, 31 (4). pp. 271-285. ISSN 1079-9893, 1532-4281

Posavec, Damir and Dorsch, Andre and Bogner, Udo and Bernhardt, Guenther and Nagl, Stefan (2011) Polyvinyl butyral nanobeads: preparation, characterization, biocompatibility and cancer cell uptake. MICROCHIMICA ACTA, 173 (3-4). pp. 391-399. ISSN 0026-3672

Puentes, Cristian Ochoa and Hoecherl, Peter and Kuehnle, Matthias and Bauer, Stefanie and Buerger, Kira and Bernhardt, Guenther and Buschauer, Armin and Koenig, Burkhard (2011) Solid phase synthesis of tariquidar-related modulators of ABC transporters preferring breast cancer resistance protein (ABCG2). BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 21 (12). pp. 3654-3657. ISSN 0960-894X, 1464-3405

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Schnell, David and Brunskole, Irena and Ladova, Katerina and Schneider, Erich H. and Igel, Patrick and Dove, Stefan and Buschauer, Armin and Seifert, Roland (2011) Expression and functional properties of canine, rat, and murine histamine H-4 receptors in Sf9 insect cells. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 383 (5). pp. 457-470. ISSN 0028-1298, 1432-1912

Seifert, Roland and Schneider, Erich H. and Dove, Stefan and Brunskole, Irena and Neumann, Detlef and Strasser, Andrea and Buschauer, Armin (2011) Paradoxical Stimulatory Effects of the "Standard" Histamine H-4-Receptor Antagonist JNJ7777120: the H-4 Receptor Joins the Club of 7 Transmembrane Domain Receptors Exhibiting Functional Selectivity. MOLECULAR PHARMACOLOGY, 79 (4). pp. 631-638. ISSN 0026-895X, 1521-0111

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Wagner, Eva and Wittmann, Hans-Joachim and Elz, Sigurd and Strasser, Andrea (2011) Mepyramine-JNJ7777120-hybrid compounds show high affinity to hH(1)R, but low affinity to hH(4)R. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 21 (21). pp. 6274-6280. ISSN 0960-894X

Weiss, Stefan and Bernhardt, Guenther and Buschauer, Armin and Koenig, Burkhard (2011) SYNTHESIS AND CHARACTERIZATION OF DMAP-MODIFIED NPY Y-1 RECEPTOR ANTAGONISTS AS ACYL-TRANSFER CATALYSTS. COLLECTION OF CZECHOSLOVAK CHEMICAL COMMUNICATIONS, 76 (6). pp. 763-780. ISSN 0010-0765

Wittmann, Hans-Joachim and Elz, Sigurd and Seifert, Roland and Strasser, Andrea (2011) N (alpha)-Methylated phenylhistamines exhibit affinity to the hH(4)R-a pharmacological and molecular modelling study. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 384 (3). pp. 287-299. ISSN 0028-1298, 1432-1912