Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer)" and Year is 2014

C

Cuboni, Serena and Devigny, Christian and Hoogeland, Bastiaan and Strasser, Andrea and Pomplun, Sebastian and Hauger, Barbara and Hoefner, Georg and Wanner, Klaus T. and Eder, Matthias and Buschauer, Armin and Holsboer, Florian and Hausch, Felix (2014) Loratadine and Analogues: Discovery and Preliminary Structure-Activity Relationship of Inhibitors of the Amino Acid Transporter B(0)AT2. JOURNAL OF MEDICINAL CHEMISTRY, 57 (22). pp. 9473-9479. ISSN 0022-2623, 1520-4804

D

Darras, Fouad H. and Pockes, Steffen and Huang, Guozhenz and Wehle, Sarah and Strasser, Andrea and Wittmann, Hans-Joachim and Nimczick, Martin and Sotriffer, Christoph A. and Decker, Michael (2014) Synthesis, Biological Evaluation, and Computational Studies of Tri- and Tetracyclic Nitrogen-Bridgehead Compounds as Potent Dual-Acting AChE Inhibitors and hH(3) Receptor Antagonists. ACS CHEMICAL NEUROSCIENCE, 5 (3). pp. 225-242. ISSN 1948-7193

F

Felixberger, J. and Strasser, A. and Tanaka, M. and Elz, S. and Bernhardt, G. and Ozawa, T. and Buschauer, A. (2014) BIASED AGONISM AT THE HISTAMINE H-1 RECEPTOR: CHIRAL HISTAPRODIFEN DERIVATIVES SHOW FUNCTIONAL SELECTIVITY FOR beta-ARRESTIN RECRUITMENT. SPRINGER BASEL AG, BASEL.

G

Geyer, Roland and Igel, Patrick and Kaske, Melanie and Elz, Sigurd and Buschauer, Armin (2014) Synthesis, SAR and selectivity of 2-acyl-and 2-cyano-1-hetarylalkyl-guanidines at the four histamine receptor subtypes: a bioisosteric approach. MEDCHEMCOMM, 5 (1). pp. 72-81. ISSN 2040-2503, 2040-2511

Geyer, Roland and Kaske, Melanie and Baumeister, Paul and Buschauer, Armin (2014) Synthesis and Functional Characterization of Imbutamine Analogs as Histamine H-3 and H-4 Receptor Ligands. ARCHIV DER PHARMAZIE, 347 (2). pp. 77-88. ISSN 0365-6233, 1521-4184

K

Kagermeier, N. and Nordemann, U. and Bernhardt, G. and Koenig, G. and Buschauer, A. (2014) DIFFERENTIAL SIGNALING PATHWAYS OF THE hH(1)R AND THE hH(2)R. SPRINGER BASEL AG, BASEL.

R

Reinartz, Michael T. and Littmann, Timo and Wainer, Irving William and Ozawa, Takeaki and Dove, Stefan and Seifert, Roland (2014) Quantifying ligand bias of enantiopure fenoterol derivatives in molecular and cellular beta(2)-adrenergic assay systems. SPRINGER, NEW YORK.

W

Wagner, Eva and Wittmann, Hans-Joachim and Elz, Sigurd and Strasser, Andrea (2014) Pharmacological profile of astemizole-derived compounds at the histamine H-1 and H-4 receptor-H-1/H-4 receptor selectivity. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 387 (3). pp. 235-250. ISSN 0028-1298, 1432-1912

Werner, Kristin and Neumann, Detlef and Buschauer, Armin and Seifert, Roland (2014) No Evidence for Histamine H-4 Receptor in Human Monocytes. JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS, 351 (3). pp. 519-526. ISSN 0022-3565, 1521-0103

Wifling, D. and Loeffel, K. and Nordemann, U. and Bernhardt, G. and Dove, S. and Seifert, R. and Buschauer, A. (2014) IN SEARCH FOR KEY AMINO ACIDS DETERMINING THE HIGH CONSTITUTIVE ACTIVITY OF THE HUMAN HISTAMINE H-4 RECEPTOR (hH(4)R). SPRINGER BASEL AG, BASEL.

Wittmann, Hans-Joachim and Seifert, Roland and Strasser, Andrea (2014) Sodium binding to hH(3)R and hH(4)R - a molecular modeling study. JOURNAL OF MOLECULAR MODELING, 20 (8): 2394. ISSN 1610-2940, 0948-5023

Wolter, Sabine and Dove, Stefan and Golombek, Marina and Schwede, Frank and Seifert, Roland (2014) N-4-monobutyryl-cCMP activates PKA RI alpha and PKA RII alpha more potently and with higher efficacy than PKG I alpha in vitro but not in vivo. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 387 (12). pp. 1163-1175. ISSN 0028-1298, 1432-1912