Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer)" and Year is 2015

B

Baumeister, Paul and Erdmann, Daniela and Biselli, Sabrina and Kagermeier, Nicole and Elz, Sigurd and Bernhardt, Guenther and Buschauer, Armin (2015) [H-3]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H-2 Receptor Antagonist. CHEMMEDCHEM, 10 (1). pp. 83-93. ISSN 1860-7179, 1860-7187

Beermann, Silke and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin and Neumann, Detlef (2015) Histamine H-1- and H-4-receptor signaling cooperatively regulate MAPK activation. BIOCHEMICAL PHARMACOLOGY, 98 (3). pp. 432-439. ISSN 0006-2952, 1873-2968

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Huber, S. and Antoni, F. and Schickaneder, C. and Schickaneder, H. and Bernhardt, G. and Buschauer, A. (2015) Stabilities of neutral and basic esters of bendamustine in plasma compared to the parent compound: Kinetic investigations by HPLC. JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 104. pp. 137-143. ISSN 0731-7085, 1873-264X

Huber, Stefan and Huettner, Johannes Philip and Hacker, Kristina and Bernhardt, Guenther and Koenig, Joerg and Buschauer, Armin (2015) Esters of Bendamustine Are by Far More Potent Cytotoxic Agents than the Parent Compound against Human Sarcoma and Carcinoma Cells. PLOS ONE, 10 (7): e0133743. ISSN 1932-6203

Huber, Stefan and Wege, Anja K. and Bernhardt, Guenther and Buschauer, Armin and Brockhoff, Gero (2015) Topotecan-induced ABCG2 expression in MCF-7 cells is associated with decreased CD24 and EpCAM expression and a loss of tumorigenicity. CYTOMETRY PART A, 87A (8). pp. 707-716. ISSN 1552-4922, 1552-4930

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Kaczor, Agnieszka A. and Guixa-Gonzalez, Ramon and Carrio, Pau and Poso, Antti and Dove, Stefan and Pastor, Manuel and Selent, Jana (2015) Multi-Component Protein - Protein Docking Based Protocol with External Scoring for Modeling Dimers of G Protein-Coupled Receptors. MOLECULAR INFORMATICS, 34 (4). pp. 246-255. ISSN 1868-1743, 1868-1751

Kagermeier, Nicole and Werner, Kristin and Keller, Max and Baumeister, Paul and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin (2015) Dimeric carbamoylguanidine-type histamine H-2 receptor ligands: A new class of potent and selective agonists. BIOORGANIC & MEDICINAL CHEMISTRY, 23 (14). pp. 3957-3969. ISSN 0968-0896, 1464-3391

Keller, Max and Schindler, Lisa and Bernhardt, Guenther and Buschauer, Armin (2015) Toward Labeled Argininamide-Type NPY Y-1 Receptor Antagonists: Identification of a Favorable Propionylation Site in BIBO3304. ARCHIV DER PHARMAZIE, 348 (6). pp. 390-398. ISSN 0365-6233, 1521-4184

Keller, Max and Traenkle, Christian and She, Xueke and Pegoli, Andrea and Bernhardt, Guenther and Buschauer, Armin and Read, Roger W. (2015) M-2 Subtype preferring dibenzodiazepinone-type muscarinic receptor ligands: Effect of chemical homo-dimerization on orthosteric (and allosteric?) binding. BIOORGANIC & MEDICINAL CHEMISTRY, 23 (14). pp. 3970-3990. ISSN 0968-0896, 1464-3391

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Orlando, Zoya and Lengers, Isabelle and Melzig, Matthias F. and Buschauer, Armin and Hensel, Andreas and Jose, Joachim (2015) Autodisplay of Human Hyaluronidase Hyal-1 on Escherichia coli and Identification of Plant-Derived Enzyme Inhibitors. MOLECULES, 20 (9). pp. 15449-15468. ISSN 1420-3049

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Reinartz, Michael T. and Kaelble, Solveig and Littmann, Timo and Ozawa, Takeaki and Dove, Stefan and Kaever, Volkhard and Wainer, Irving W. and Seifert, Roland (2015) Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the beta(2)-adrenoceptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 388 (1). pp. 51-65. ISSN 0028-1298, 1432-1912

Rothenhoefer, Martin and Grundmann, Marco and Bernhardt, Guenther and Matysik, Frank-Michael and Buschauer, Armin (2015) High performance anion exchange chromatography with pulsed amperometric detection (HPAEC-PAD) for the sensitive determination of hyaluronan oligosaccharides. JOURNAL OF CHROMATOGRAPHY B-ANALYTICAL TECHNOLOGIES IN THE BIOMEDICAL AND LIFE SCIENCES, 988. pp. 106-115. ISSN 1570-0232, 1873-376X

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Slattery, David A. and Naik, Roshan R. and Grund, Thomas and Yen, Yi-Chun and Sartori, Simone B. and Fuechsl, Andrea and Finger, Beate C. and Elfving, Betina and Nordemann, Uwe and Guerrini, Remo and Calo, Girolamo and Wegener, Gregers and Mathe, Aleksander A. and Singewald, Nicolas and Czibere, Ludwig and Landgraf, Rainer and Neumann, Inga D. (2015) Selective Breeding for High Anxiety Introduces a Synonymous SNP That Increases Neuropeptide S Receptor Activity. JOURNAL OF NEUROSCIENCE, 35 (11). pp. 4599-4613. ISSN 0270-6474

Strasser, Andrea and Wittmann, Hans-Joachim and Schneider, Erich H. and Seifert, Roland (2015) Modulation of GPCRs by monovalent cations and anions. SPRINGER, NEW YORK.

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Untergehrer, Monika and Buecherl, Daniel and Wittmann, Hans-Joachim and Strasser, Andrea and Heilmann, Joerg and Juergenliemk, Guido (2015) Structure-Dependent Deconjugation of Flavonoid Glucuronides by Human beta-Glucuronidase - In Vitro and In Silico Analyses. PLANTA MEDICA, 81 (12-13). pp. 1182-1189. ISSN 0032-0943, 1439-0221

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Werner, Kristin and Kaelble, Solveig and Wolter, Sabine and Schneider, Erich H. and Buschauer, Armin and Neumann, Detlef and Seifert, Roland (2015) Flow cytometric analysis with a fluorescently labeled formyl peptide receptor ligand as a new method to study the pharmacological profile of the histamine H-2 receptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 388 (10). pp. 1039-1052. ISSN 0028-1298, 1432-1912

Wifling, David and Bernhardt, Guenther and Dove, Stefan and Buschauer, Armin (2015) The Extracellular Loop 2 (ECL2) of the Human Histamine H-4 Receptor Substantially Contributes to Ligand Binding and Constitutive Activity. PLOS ONE, 10 (1): e0117185. ISSN 1932-6203

Wittmann, Hans-Joachim and Strasser, Andrea (2015) Binding pathway of histamine to the hH(4)R, observed by unconstrained molecular dynamics. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 25 (6). pp. 1259-1268. ISSN 0960-894X, 1464-3405