Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer)" and Year is 2020

A

Andreev, Stanislav and Pantsar, Tatu and El-Gokha, Ahmed and Ansideri, Francesco and Kudolo, Mark and Anton, Debora Bublitz and Sita, Giulia and Romasco, Jenny and Geibel, Christian and Laemmerhofer, Michael and Goettert, Marcia Ines and Tarozzi, Andrea and Laufer, Stefan A. and Koch, Pierre (2020) Discovery and Evaluation of Enantiopure 9H-pyrimido[4,5-b]indoles as Nanomolar GSK-3 beta Inhibitors with Improved Metabolic Stability. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (21): 7823. ISSN 1422-0067

Antoni, Frauke and Bause, Manuel and Scholler, Matthias and Bauer, Stefanie and Stark, Simone A. and Jackson, Scott M. and Manolaridis, Ioannis and Locher, Kaspar P. and Koenig, Burkhard and Buschauer, Armin and Bernhardt, Guenther (2020) Tariquidar-related triazoles as potent, selective and stable inhibitors of ABCG2 (BCRP). EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 191: 112133. ISSN 0223-5234, 1768-3254

B

Bartole, Edith and Graetz, Lukas and Littmann, Timo and Wifling, David and Seibel, Ulla and Buschauer, Armin and Bernhardt, Guenther (2020) UR-DEBa242: A Py-5-Labeled Fluorescent Multipurpose Probe for Investigations on the Histamine H-3 and H-4 Receptors. JOURNAL OF MEDICINAL CHEMISTRY, 63 (10). pp. 5297-5311. ISSN 0022-2623, 1520-4804

Biselli, Sabrina and Alencastre, Ines and Tropmann, Katharina and Erdmann, Daniela and Chen, Mengya and Littmann, Timo and Maia, Andre F. and Gomez-Lazaro, Maria and Tanaka, Miho and Ozawa, Takeaki and Keller, Max and Lamghari, Meriem and Buschauer, Armin and Bernhardt, Guenther (2020) Fluorescent H-2 Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications. ACS MEDICINAL CHEMISTRY LETTERS, 11 (8). pp. 1521-1528. ISSN 1948-5875

Buschmann, Jonas and Seiler, Theresa and Bernhardt, Guenther and Keller, Max and Wifling, David (2020) Argininamide-type neuropeptide Y Y-1 receptor antagonists: the nature of N-omega-carbamoyl substituents determines Y1R binding mode and affinity. RSC MEDICINAL CHEMISTRY, 11 (2). pp. 274-282. ISSN 2632-8682

F

Forster, Lisa and Graetz, Lukas and Moennich, Denise and Bernhardt, Guenther and Pockes, Steffen (2020) A Split Luciferase Complementation Assay for the Quantification of beta-Arrestin2 Recruitment to Dopamine D-2-Like Receptors. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (17): 6103. ISSN 1422-0067

G

Gruber, Corinna G. and Pegoli, Andrea and Mueller, Christoph and Graetz, Lukas and She, Xueke and Keller, Max (2020) Differently fluorescence-labelled dibenzodiazepinone-type muscarinic acetylcholine receptor ligands with high M2R affinity. RSC MEDICINAL CHEMISTRY, 11 (7). pp. 823-832. ISSN 2632-8682

H

Hoering, Carina and Seibel, Ulla and Littmann, Timo and Graetz, Lukas and Strasser, Andrea and Bernhardt, Guenther (2020) A MiniG Protein Recruitment Assay for the Histamine Receptor Family to Functionally Characterize Histamine Receptor Ligands. In: Annual Meeting on Experimental Biology, APR 04-07, 2020, San Diego, CA.

Horing, Carina and Seibel, Ulla and Tropmann, Katharina and Gratz, Lukas and Monnich, Denise and Pitzl, Sebastian and Bernhardt, Gunther and Pockes, Steffen and Strasser, Andrea (2020) A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 21 (22): 8440. ISSN 1422-0067

K

Konieczny, Adam and Braun, Diana and Wifling, David and Bernhardt, Guenther and Keller, Max (2020) Oligopeptides as Neuropeptide Y Y-4 Receptor Ligands: Identification of a High-Affinity Tetrapeptide Agonist and a Hexapeptide Antagonist. JOURNAL OF MEDICINAL CHEMISTRY, 63 (15). pp. 8198-8215. ISSN 0022-2623, 1520-4804

S

She, Xueke and Pegoli, Andrea and Gruber, Corinna G. and Wifling, David and Carpenter, Jessica and Huebner, Harald and Chen, Mengya and Wan, Jianfei and Bernhardt, Guenther and Gmeiner, Peter and Holliday, Nicholas D. and Keller, Max (2020) Red-Emitting Dibenzodiazepinone Derivatives as Fluorescent Dualsteric Probes for the Muscarinic Acetylcholine M-2 Receptor. JOURNAL OF MEDICINAL CHEMISTRY, 63 (8). pp. 4133-4154. ISSN 0022-2623, 1520-4804