Items where Division is "Chemistry and Pharmacy > Institute of Pharmacy > Pharmaceutical/Medicinal Chemistry II (Prof. Buschauer)" and Year is 2021

A

Antoni, Frauke and Wifling, David and Bernhardt, Guenther (2021) Water-soluble inhibitors of ABCG2 (BCRP) - A fragment-based and computational approach. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 210: 112958. ISSN 0223-5234, 1768-3254

B

Biselli, Sabrina and Bresinsky, Merlin and Tropmann, Katharina and Forster, Lisa and Honisch, Claudia and Buschauer, Armin and Bernhardt, Gunther and Pockes, Steffen (2021) Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H2R and D3R. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 214: 113190. ISSN 0223-5234, 1768-3254

E

Eitel, Michael and Zinad, Dhafer S. and Schollmeyer, Dieter and Gross, Harald and Koch, Pierre (2021) Selective mono-de-O-acetylation of the per-O-acetylated brasilicardin carbohydrate side chain. CARBOHYDRATE RESEARCH, 504: 108312. ISSN 0008-6215, 1873-426X

F

Forster, L. and Graetz, L. and Moennich, D. and Bernhardt, G. and Pockes, S. (2021) A split luciferase complementation assay for the quantification of beta-arrestin2 recruitment to dopamine D-2-like receptors. In: 87th Annual Meeting of the German Society for Experimental and Clinical Pharmacology and Toxicology (DGPT), March 01-03, 2021, Digital.

H

Hoering, Carina and Conrad, Marcus and Soldner, Christian A. and Wang, Jinan and Sticht, Heinrich and Strasser, Andrea and Miao, Yinglong (2021) Specific Engineered G Protein Coupling to Histamine Receptors Revealed from Cellular Assay Experiments and Accelerated Molecular Dynamics Simulations. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, 22 (18): 10047. ISSN , 1422-0067

Hoffmeister, Helen and Fuchs, Andreas and Komives, Elizabeth and Groebner-Ferreira, Regina and Strobl, Laura and Nazet, Julian and Heizinger, Leonhard and Merkl, Rainer and Dove, Stefan and Laengst, Gernot (2021) Sequence and functional differences in the ATPase domains of CHD3 and SNF2H promise potential for selective regulability and drugability. FEBS JOURNAL, 288 (13). pp. 4000-4023. ISSN 1742-464X, 1742-4658

K

Konieczny, Adam and Conrad, Marcus and Ertl, Fabian J. and Gleixner, Jakob and Gattor, Albert O. and Graetz, Lukas and Schmidt, Maximilian F. and Neu, Eduard and Horn, Anselm H. C. and Wifling, David and Gmeiner, Peter and Clark, Timothy and Sticht, Heinrich and Keller, Max (2021) N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y-4 Receptor Ligands Results in Picomolar Binding Constants. JOURNAL OF MEDICINAL CHEMISTRY, 64 (22). pp. 16746-16769. ISSN 0022-2623, 1520-4804

R

Reynders, Martin and Chaikuad, Apirat and Berger, Benedict-Tilman and Bauer, Katharina and Koch, Pierre and Laufer, Stefan and Knapp, Stefan and Trauner, Dirk (2021) Controlling the Covalent Reactivity of a Kinase Inhibitor with Light. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 60 (37). pp. 20178-20183. ISSN 1433-7851, 1521-3773

T

Tropmann, Katharina and Bresinsky, Merlin and Forster, Lisa and Moennich, Denise and Buschauer, Armin and Wittmann, Hans-Joachim and Huebner, Harald and Gmeiner, Peter and Pockes, Steffen and Strasser, Andrea (2021) Abolishing Dopamine D-2long/D-3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H-2 Receptor Agonists. JOURNAL OF MEDICINAL CHEMISTRY, 64 (12). pp. 8684-8709. ISSN 0022-2623, 1520-4804

W

Weinhart, Corinna G. and Wifling, David and Schmidt, Maximilian F. and Neu, Eduard and Hoering, Carina and Clark, Timothy and Gmeiner, Peter and Keller, Max (2021) Dibenzodiazepinone-type muscarinic receptor antagonists conjugated to basic peptides: Impact of the linker moiety and unnatural amino acids on M2R selectivity. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 213: 113159. ISSN 0223-5234, 1768-3254