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A

Aiglstorfer, Iris and Hendrich, Ingo and Moser, Christiane and Bernhardt, Günther and Dove, Stefan and Buschauer, Armin (2000) Structure-activity relationships of neuropeptide YY1 receptor antagonists related to BIBP 3226. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 10 (14). pp. 1597-1600. ISSN 0960-894X

B

Barbic, M. and Willer, E. A. and Rothenhoefer, M. and Heilmann, J. and Fuerst, R. and Juergenliemk, G. (2013) Spirostanol saponins and esculin from Rusci rhizoma reduce the thrombin-induced hyperpermeability of endothelial cells. PHYTOCHEMISTRY, 90. pp. 106-113. ISSN 0031-9422

Beermann, Silke and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin and Neumann, Detlef (2015) Histamine H-1- and H-4-receptor signaling cooperatively regulate MAPK activation. BIOCHEMICAL PHARMACOLOGY, 98 (3). pp. 432-439. ISSN 0006-2952, 1873-2968

Bouchal, Jan and Kolar, Zdenek and Mad'arova, Jana and Hlobilkova, Alice and von Angerer, Erwin (2002) The effects of natural ligands of hormone receptors and their antagonists on telomerase activity in the androgen sensitive prostatic cancer cell line LNCaP. BIOCHEMICAL PHARMACOLOGY, 63 (6): PII S0006-. pp. 1177-1181. ISSN 0006-2952

Brennauer, Albert and Keller, Max and Freund, Matthias and Bernhardt, Guenther and Buschauer, Armin (2007) Decomposition of 1-(omega-aminoalkanoyl)guanidines under alkaline conditions. TETRAHEDRON LETTERS, 48 (39). pp. 6996-6999. ISSN 0040-4039

G

Ghorai, Prasanta and Kraus, Anja and Birnkammer, Tobias and Geyer, Roland and Bernhardt, Guenther and Dove, Stefan and Seifert, Roland and Elz, Sigurd and Buschauer, Armin (2010) Chiral N-G-acylated hetarylpropylguanidine-type histamine H-2 receptor agonists do not show significant stereoselectivity. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 20 (10). pp. 3173-3176. ISSN 0960-894X

I

Igel, Patrick and Dove, Stefan and Buschauer, Armin (2010) Histamine H-4 receptor agonists. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 20 (24). pp. 7191-7199. ISSN 0960-894X, 1464-3405

K

Kagermeier, Nicole and Werner, Kristin and Keller, Max and Baumeister, Paul and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin (2015) Dimeric carbamoylguanidine-type histamine H-2 receptor ligands: A new class of potent and selective agonists. BIOORGANIC & MEDICINAL CHEMISTRY, 23 (14). pp. 3957-3969. ISSN 0968-0896, 1464-3391

Katsouri, Ilektra Petrina and Vandervelpen, Ebert Vinciane G. and Gattor, Albert Owusu and Engelbeen, Sarah and El Sayed, Abdulrahman and Seitaj, Klejdia and Becerra, Eduardo Daniel Morales and Vanderheyden, Patrick M. L. (2022) Complex FFA1 receptor (in)dependent modulation of calcium signaling by free fatty acids. BIOCHEMICAL PHARMACOLOGY, 202: 115150. ISSN 0006-2952, 1873-2968

Kaufmann, Doris and Pojarova, Michaela and Vogel, Susanne and Liebl, Renate and Gastpar, Robert and Gross, Dietmar and Nishino, Tsuyuki and Pfaller, Tobias and von Angerer, Erwin (2007) Antimitotic activities of 2-phenylindole-3-carbaldehydes in human breast cancer cells. BIOORGANIC & MEDICINAL CHEMISTRY, 15 (15). pp. 5122-5136. ISSN 0968-0896, 1464-3391

Keller, Max and Erdmann, Daniela and Pop, Nathalie and Pluym, Nikola and Teng, Shangjun and Bernhardt, Guenther and Buschauer, Armin (2011) Red-fluorescent argininamide-type NPY Y-1 receptor antagonists as pharmacological tools. BIOORGANIC & MEDICINAL CHEMISTRY, 19 (9). pp. 2859-2878. ISSN 0968-0896, 1464-3391

Keller, Max and Kaske, Melanie and Holzammer, Tobias and Bernhardt, Guenther and Buschauer, Armin (2013) Dimeric argininamide-type neuropeptide Y receptor antagonists: Chiral discrimination between Y-1 and Y-4 receptors. BIOORGANIC & MEDICINAL CHEMISTRY, 21 (21). pp. 6303-6322. ISSN 0968-0896, 1464-3391

Keller, Max and Traenkle, Christian and She, Xueke and Pegoli, Andrea and Bernhardt, Guenther and Buschauer, Armin and Read, Roger W. (2015) M-2 Subtype preferring dibenzodiazepinone-type muscarinic receptor ligands: Effect of chemical homo-dimerization on orthosteric (and allosteric?) binding. BIOORGANIC & MEDICINAL CHEMISTRY, 23 (14). pp. 3970-3990. ISSN 0968-0896, 1464-3391

Knieps, Sebastian and Michel, Martin C. and Dove, Stefan and Buschauer, Armin (1995) Non-peptide neuropeptide y antagonists derived from the histamine H2 agonist arpromidine: Role of the guanidine group. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 5 (18). pp. 2065-2070. ISSN 0960-894X, 1464-3405

L

Lazewska, Dorota and Mogilski, Szczepan and Hagenow, Stefanie and Kuder, Kamil and Gluch-Lutwin, Monika and Siwek, Agata and Wiecek, Malgorzata and Kaleta, Maria and Seibel, Ulla and Buschauer, Armin and Filipek, Barbara and Stark, Holger and Kiec-Kononowicz, Katarzyna (2019) Alkyl derivatives of 1,3,5-triazine as histamine H-4 receptor ligands. BIOORGANIC & MEDICINAL CHEMISTRY, 27 (7). pp. 1254-1262. ISSN 0968-0896, 1464-3391

Li, Liantao and Kracht, Julia and Peng, Shiqi and Bernhardt, Günther and Buschauer, Armin (2003) Synthesis and pharmacological activity of fluorescent histamine H-1 receptor antagonists related to mepyramine. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 13 (7). pp. 1245-1248. ISSN 0960-894X

Loeber, Stefan and Huebner, Harald and Buschauer, Armin and Sanna, Fabrizio and Argiolas, Antonio and Melis, Maria Rosaria and Gmeiner, Peter (2012) Novel azulene derivatives for the treatment of erectile dysfunction. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 22 (23). pp. 7151-7154. ISSN 0960-894X

P

Pojarova, Michaela and Kaufmann, Doris and Gastpar, Robert and Nishino, Tsuyuki and Reszka, Przemyslaw and Bednarski, Patrick J. and von Angerer, Erwin (2007) [(2-Phenylindol-3-yl)methylene]propanedinitriles inhibit the growth of breast cancer cells by cell cycle arrest in G(2)/M phase and apoptosis. BIOORGANIC & MEDICINAL CHEMISTRY, 15 (23). pp. 7368-7379. ISSN 0968-0896, 1464-3391

Puentes, Cristian Ochoa and Hoecherl, Peter and Kuehnle, Matthias and Bauer, Stefanie and Buerger, Kira and Bernhardt, Guenther and Buschauer, Armin and Koenig, Burkhard (2011) Solid phase synthesis of tariquidar-related modulators of ABC transporters preferring breast cancer resistance protein (ABCG2). BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 21 (12). pp. 3654-3657. ISSN 0960-894X, 1464-3405

R

Reher, Till M. and Brunskole, Irena and Neumann, Detlef and Seifert, Roland (2012) Evidence for ligand-specific conformations of the histamine H-2-receptor in human eosinophils and neutrophils. BIOCHEMICAL PHARMACOLOGY, 84 (9). pp. 1174-1185. ISSN 0006-2952

Reher, Till M. and Neumann, Detlef and Buschauer, Armin and Seifert, Roland (2012) Incomplete activation of human eosinophils via the histamine H-4-receptor: Evidence for ligand-specific receptor conformations. BIOCHEMICAL PHARMACOLOGY, 84 (2). pp. 192-203. ISSN 0006-2952, 1873-2968

S

Schnell, David and Strasser, Andrea and Seifert, Roland (2010) Comparison of the pharmacological properties of human and rat histamine H-3-receptors. BIOCHEMICAL PHARMACOLOGY, 80 (9). pp. 1437-1449. ISSN 0006-2952

Seifert, Roland and Dove, Stefan (2013) Inhibitors of Bacillus anthracis edema factor. PERGAMON-ELSEVIER SCIENCE LTD, OXFORD.

Spickenreither, Martin and Braun, Stephan and Bernhardt, Guenther and Dove, Stefan and Buschauer, Armin (2006) Novel 6-O-acylated vitamin C derivatives as hyaluronidase inhibitors with selectivity for bacterial lyases. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 16 (20). pp. 5313-5316. ISSN 0960-894X

W

Wabnitz, Tobias C. and Rizzo, Simona and Goette, Carsten and Buschauer, Armin and Benincori, Tiziana and Reiser, Oliver (2006) Enantioselective hydrogenation of diaryl-substituted alpha,beta-unsaturated nitriles. TETRAHEDRON LETTERS, 47 (22). pp. 3733-3736. ISSN 0040-4039

Wagner, Eva and Wittmann, Hans-Joachim and Elz, Sigurd and Strasser, Andrea (2011) Mepyramine-JNJ7777120-hybrid compounds show high affinity to hH(1)R, but low affinity to hH(4)R. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 21 (21). pp. 6274-6280. ISSN 0960-894X

Walter, Georg and Liebl, Renate and von Angerer, Erwin (2004) Synthesis and biological evaluation of stilbene-based pure estrogen antagonists. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 14 (18). pp. 4659-4663. ISSN 0960-894X, 1464-3405

Weiss, Stefan and Keller, Max and Bernhardt, Guenther and Buschauer, Armin and Koenig, Burkhard (2008) Modular synthesis of non-peptidic bivalent NPY Y-1 receptor antagonists. BIOORGANIC & MEDICINAL CHEMISTRY, 16 (22). pp. 9858-9866. ISSN 0968-0896

Weiss, Stefan and Keller, Max and Bernhardt, Guenther and Buschauer, Armin and Koenig, Burkhard (2010) N-G-Acyl-argininamides as NPY Y-1 receptor antagonists: Influence of structurally diverse acyl substituents on stability and affinity. BIOORGANIC & MEDICINAL CHEMISTRY, 18 (17). pp. 6292-6304. ISSN 0968-0896

Wittmann, Hans-Joachim and Strasser, Andrea (2015) Binding pathway of histamine to the hH(4)R, observed by unconstrained molecular dynamics. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 25 (6). pp. 1259-1268. ISSN 0960-894X, 1464-3405

X

Xie, Sheng-Xue and Petrache, Georgiana and Schneider, Erich and Ye, Qi-Zhuang and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin (2006) Synthesis and pharmacological characterization of novel fluorescent histamine H-2-receptor ligands derived from aminopotentidine. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 16 (15). pp. 3886-3890. ISSN 0960-894X