Browse by ["viewname_eprint_publisher" not defined]

B

Beermann, Silke and Bernhardt, Guenther and Seifert, Roland and Buschauer, Armin and Neumann, Detlef (2015) Histamine H-1- and H-4-receptor signaling cooperatively regulate MAPK activation. BIOCHEMICAL PHARMACOLOGY, 98 (3). pp. 432-439. ISSN 0006-2952, 1873-2968

Biberger, C. and von Angerer, Erwin (1998) 1-benzyl-2-phenylindole- and 1,2-diphenylindole-based antiestrogens. Estimation of agonist and antagonist activities in transfection assays. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 64 (5-6). pp. 277-285. ISSN 0960-0760,

Biberger, C. and von Angerer, Erwin (1996) 2-phenylindoles with sulfur containing side chains. Estrogen receptor affinity, antiestrogenic potency, and antitumor activity. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 58 (1). pp. 31-43. ISSN 0960-0760

C

Chen, Xinyu and Tikhonova, Irina G. and Decker, Michael (2011) Probing the mid-gorge of cholinesterases with spacer-modified bivalent quinazolinimines leads to highly potent and selective butyrylcholinesterase inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY, 19 (3). pp. 1222-1235. ISSN 0968-0896, 1464-3391

D

Darras, Fouad H. and Kling, Beata and Sawatzky, Edgar and Heilmann, Joerg and Decker, Michael (2014) Cyclic acyl guanidines bearing carbamate moieties allow potent and dirigible cholinesterase inhibition of either acetyl- or butyrylcholinesterase. BIOORGANIC & MEDICINAL CHEMISTRY, 22 (17). pp. 5020-5034. ISSN 0968-0896, 1464-3391

Darras, Fouad H. and Wehle, Sarah and Huang, Guozheng and Sotriffer, Christoph A. and Decker, Michael (2014) Amine substitution of quinazolinones leads to selective nanomolar AChE inhibitors with 'inverted' binding mode. BIOORGANIC & MEDICINAL CHEMISTRY, 22 (17). pp. 4867-4881. ISSN 0968-0896, 1464-3391

G

Golob, Thomas and Liebl, Renate and von Angerer, Erwin (2002) Sulfamoyloxy-substituted 2-phenylindoles: Antiestrogen-based inhibitors of the steroid sulfatase in human breast cancer cells. BIOORGANIC & MEDICINAL CHEMISTRY, 10 (12). pp. 3941-3953. ISSN 0968-0896

H

Hafner, F. and Holler, Eggehard and von Angerer, E. (1996) Effect of growth factors on estrogen receptor mediated gene expression. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 58 (4). pp. 385-393. ISSN 0960-0760

Hammer, Sebastian G. and Gobleder, Susanne and Naporra, Franziska and Wittmann, Hans-Joachim and Elz, Sigurd and Heinrich, Markus R. and Strasser, Andrea (2016) 2,4-Diaminopyrimidines as dual ligands at the histamine H-1 and H-4 receptor-H-1/H-4-receptor selectivity. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 26 (2). pp. 292-300. ISSN 0960-894X, 1464-3405

K

Kaufmann, Doris and Pojarova, Michaela and Vogel, Susanne and Liebl, Renate and Gastpar, Robert and Gross, Dietmar and Nishino, Tsuyuki and Pfaller, Tobias and von Angerer, Erwin (2007) Antimitotic activities of 2-phenylindole-3-carbaldehydes in human breast cancer cells. BIOORGANIC & MEDICINAL CHEMISTRY, 15 (15). pp. 5122-5136. ISSN 0968-0896, 1464-3391

L

Lazewska, Dorota and Mogilski, Szczepan and Hagenow, Stefanie and Kuder, Kamil and Gluch-Lutwin, Monika and Siwek, Agata and Wiecek, Malgorzata and Kaleta, Maria and Seibel, Ulla and Buschauer, Armin and Filipek, Barbara and Stark, Holger and Kiec-Kononowicz, Katarzyna (2019) Alkyl derivatives of 1,3,5-triazine as histamine H-4 receptor ligands. BIOORGANIC & MEDICINAL CHEMISTRY, 27 (7). pp. 1254-1262. ISSN 0968-0896, 1464-3391

Luebker, Carolin and Urbauer, Ramona J. Bieber and Moskovitz, Jackob and Dove, Stefan and Weisemann, Jasmin and Fedorova, Maria and Urbauer, Jeffrey L. and Seifert, Roland (2015) Membranous adenylyl cyclase 1 activation is regulated by oxidation of N- and C-terminal methionine residues in calmodulin. BIOCHEMICAL PHARMACOLOGY, 93 (2). pp. 196-209. ISSN 0006-2952, 1873-2968

M

Mathioudaki, Angeliki and Berzesta, Ariola and Kypriotakis, Zacharias and Skaltsa, Helen and Heilmann, Joerg (2018) Phenolic metabolites from Hypericum kelleri BALD., an endemic species of Crete (Greece). PHYTOCHEMISTRY, 146. pp. 1-7. ISSN 0031-9422

Müller, Klaus and Gawlik, Ingo (1996) Inactivation of mouse epidermal 12-lipoxygenase by anthralin - Implications for the role of oxygen radicals. BIOCHEMICAL PHARMACOLOGY, 51 (9). pp. 1173-1179. ISSN 0006-2952, 1873-2968

Müller, Klaus and Gawlik, Ingo (1995) Novel 10-substituted antipsoriatic anthrones as inhibitors of epidermal 12-lipoxygenase and lipid peroxidation in membranes. BIOCHEMICAL PHARMACOLOGY, 50 (12). pp. 2077-2083. ISSN 0006-2952, 1873-2968

N

Nguyen, Le-Thu T. and Nguyen, Hieu T. and Barbic, Matej and Brunner, Gabi and Heilmann, Joerg and Pham, Hung D. and Nguyen, Duc M. and Nguyen, Lien-Hoa D. (2012) Polyisoprenylated acylphloroglucinols and a polyisoprenylated tetracyclic xanthone from the bark of Calophyllum thorelii. TETRAHEDRON LETTERS, 53 (34). pp. 4487-4493. ISSN 0040-4039

R

Radons, Juergen and Falk, Werner and Dove, Stefan (2015) Identification of critical regions within the TIR domain of IL-1 receptor type I. INTERNATIONAL JOURNAL OF BIOCHEMISTRY & CELL BIOLOGY, 68. pp. 15-20. ISSN 1357-2725, 1878-5875

Reher, Till M. and Brunskole, Irena and Neumann, Detlef and Seifert, Roland (2012) Evidence for ligand-specific conformations of the histamine H-2-receptor in human eosinophils and neutrophils. BIOCHEMICAL PHARMACOLOGY, 84 (9). pp. 1174-1185. ISSN 0006-2952

Rodrigues, Paula C. A. and Beyer, Ulrich and Schumacher, Peter and Roth, Thomas and Fiebig, Heinz H. and Unger, Clemens and Messori, Luigi and Orioli, Pierluigi and Paper, Dietrich H. and Muelhaupt, Rolf and Kratz, Felix (1999) Acid-sensitive polyethylene glycol conjugates of doxorubicin: Preparation, in vitro efficacy and intracellular distribution. BIOORGANIC & MEDICINAL CHEMISTRY, 7 (11). pp. 2517-2524. ISSN 0968-0896,

S

Sadek, Bassem and Khan, Nadia and Darras, Fouad H. and Pockes, Steffen and Decker, Michael (2016) The dual-acting AChE inhibitor and H-3 receptor antagonist UW-MD-72 reverses amnesia induced by scopolamine or dizocilpine in passive avoidance paradigm in rats. PHYSIOLOGY & BEHAVIOR, 165. pp. 383-391. ISSN 0031-9384

Sander, Kerstin and Kottke, Tim and Tanrikulu, Yusuf and Proschak, Ewgenij and Weizel, Lilia and Schneider, Erich H. and Seifert, Roland and Schneider, Gisbert and Stark, Holger (2009) 2,4-Diaminopyrimidines as histamine H-4 receptor ligands-Scaffold optimization and pharmacological characterization. BIOORGANIC & MEDICINAL CHEMISTRY, 17 (20). pp. 7186-7196. ISSN 0968-0896, 1464-3391

Schmidt, Sebastian and Juergenliemk, Guido and Skaltsa, Helen and Heilmann, Joerg (2012) Phloroglucinol derivatives from Hypericum empetrifolium with antiproliferative activity on endothelial cells. PHYTOCHEMISTRY, 77. pp. 218-225. ISSN 0031-9422

Schwindl, Sebastian and Kraus, Birgit and Heilmann, Joerg (2019) Secondary metabolites from the leaves of Juglans regia L. BIOCHEMICAL SYSTEMATICS AND ECOLOGY, 83. pp. 130-136. ISSN 0305-1978, 1873-2925

T

Tropmann, Katharina and Seibel-Ehlert, Ulla and Littmann, Timo and Strasser, Andrea (2021) Shining light on the histamine H-2 receptor: Synthesis of carbamoylguanidine-type agonists as a pharmacological tool to study internalization. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 52: 128388. ISSN 0960-894X, 1464-3405

V

Vogel, Susanne and Kaufmann, Doris and Pojarova, Michaela and Mueller, Christine and Pfaller, Tobias and Kuehne, Sybille and Bednarski, Patrick J. and von Angerer, Erwin (2008) Aroyl hydrazones of 2-phenylindole-3-carbaldehydes as novel antimitotic agents. BIOORGANIC & MEDICINAL CHEMISTRY, 16 (12). pp. 6436-6447. ISSN 0968-0896

W

Walter, Georg and Liebl, Renate and von Angerer, Erwin (2004) 2-Phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells. JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 88 (4-5). pp. 409-420. ISSN 0960-0760

Weiss, Stefan and Keller, Max and Bernhardt, Guenther and Buschauer, Armin and Koenig, Burkhard (2008) Modular synthesis of non-peptidic bivalent NPY Y-1 receptor antagonists. BIOORGANIC & MEDICINAL CHEMISTRY, 16 (22). pp. 9858-9866. ISSN 0968-0896

Wiesneth, Stefan and Aas, Gregor and Heilmann, Joerg and Juergenliemk, Guido (2018) Investigation of the flavan-3-ol patterns in willow species during one growing-season. PHYTOCHEMISTRY, 145. pp. 26-39. ISSN 0031-9422

Wittmann, Hans-Joachim and Seifert, Roland and Strasser, Andrea (2011) Influence of the N-terminus and the E2-loop onto the binding kinetics of the antagonist mepyramine and the partial agonist phenoprodifen to H1R. BIOCHEMICAL PHARMACOLOGY, 82 (12). pp. 1910-1918. ISSN 0006-2952