Browse by ["viewname_eprint_publisher" not defined]

A

Appl, H. and Holzammer, T. and Dove, S. and Seifert, R. (2010) Interaction of antipsychotic and antidepressant drugs with the four histamine receptor subtypes. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 381 (1Suppl). p. 11. ISSN 0028-1298

B

Banjarnahor, Sofna and Scherpinski, Lorenz A. and Keller, Max and Koenig, Joerg and Maas, Renke (2025) Differential uptake of arginine derivatives by the human heteromeric amino acid transporter b<SUP>0,+</SUP>AT-rBAT (SLC7A9-SLC3A1). NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 398 (4). pp. 4419-4434. ISSN 0028-1298, 1432-1912

Brunskole, I. and Buschauer, A. and Kaelble, S. and Burhenne, H. and Seifert, R. (2012) Dissociations in the effects of beta(2)-adrenergic receptor agonists on cAMP formation and superoxide production in human neutrophils. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 385 (1Suppl). S16. ISSN 0028-1298

Brunskole, I. and Strasser, A. and Buschauer, A. and Seifert, R. (2010) Contribution of extracellular domains to ligand-receptor interactions at the human histamine H-4-receptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 381 (1Suppl). p. 13. ISSN 0028-1298

Brunskole, Irena and Strasser, Andrea and Seifert, Roland and Buschauer, Armin (2011) Role of the second and third extracellular loops of the histamine H-4 receptor in receptor activation. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 384 (3). pp. 301-317. ISSN 0028-1298

E

Elz, Sigurd and Paraschiv, G.-I. and Patil, R. and Kunze, M. and Striegl, B. and Sunel, V. and Cecal, A. and Buschauer, Armin and Reiser, Oliver (2005) New side-chain modified histamine derivatives as ligands for histamine H-1-receptors. In: 46th Spring Meeting of the Deutsche Gesellschaft fuer Experimentelle und Klinische Pharmakologie und Toxikologie, March 15-17, 2005, Mainz, Germany.

F

Forster, L. and Buschauer, A. and Bernhardt, G. (2019) Investigation of GPCR-beta-arrestin interactions using a split-luciferase complementation assay: Application to the D-2long and D-3 receptor. SPRINGER, NEW YORK.

Forster, L. and Graetz, L. and Moennich, D. and Bernhardt, G. and Pockes, S. (2021) A split luciferase complementation assay for the quantification of beta-arrestin2 recruitment to dopamine D-2-like receptors. In: 87th Annual Meeting of the German Society for Experimental and Clinical Pharmacology and Toxicology (DGPT), March 01-03, 2021, Digital.

G

Graetz, L. and Littmann, T. and Bartole, E. and Biselli, S. and Pegoli, A. and Keller, M. and Buschauer, A. and Bernhardt, G. (2019) A BRET-based assay to determine the binding of ligands to GPCRs using pyrylium-labeled fluorescent tracers. SPRINGER, NEW YORK.

Gross, Dietmar and Bernhardt, Gunther and Buschauer, Armin (2006) Platelet-derived growth factor receptor independent proliferation of human glioblastoma cells: selective tyrosine kinase inhibitors lack antiproliferative activity. JOURNAL OF CANCER RESEARCH AND CLINICAL ONCOLOGY, 132 (9). pp. 589-599. ISSN 0171-5216

H

Hoering, C. and Graetz, L. and Littmann, T. and Buschauer, A. and Bernhardt, G. and Strasser, A. (2019) Mini G protein recruitment as an approach to the functional characterization of histamine receptor ligands. SPRINGER, NEW YORK.

Hofinger, Edith S. A. and Hoechstetter, Julia and Oettl, Martin and Bernhardt, Guenther and Buschauer, Armin (2008) Isoenzyme-specific differences in the degradation of hyaluronic acid by mammalian-type hyaluronidases. GLYCOCONJUGATE JOURNAL, 25 (2). pp. 101-109. ISSN 0282-0080, 1573-4986

Hubensack, Martina and Mueller, Christine and Hoecherl, Peter and Fellner, Stephan and Spruss, Thilo and Bernhardt, Guenther and Buschauer, Armin (2008) Effect of the ABCB1 modulators elacridar and tariquidar on the distribution of paclitaxel in nude mice. JOURNAL OF CANCER RESEARCH AND CLINICAL ONCOLOGY, 134 (5). pp. 597-607. ISSN 0171-5216

M

Mueller, Christine and Gross, Dietmar and Sarli, Vasiliki and Gartner, Michael and Giannis, Athanassios and Bernhardt, Guenther and Buschauer, Armin (2007) Inhibitors of kinesin Eg5: antiproliferative activity of monastrol analogues against human glioblastoma cells. CANCER CHEMOTHERAPY AND PHARMACOLOGY, 59 (2). pp. 157-164. ISSN 0344-5704

P

Pockes, S. and Buschauer, A. and Elz, S. (2016) In-vitro-pharmacology and structure-activity relationships of derivatives of imidazolylpropylguanidine (SK&F-91,486) at histamine receptors (hH(1,2,3,4)R and gpH(1,2)R). SPRINGER, NEW YORK.

Preuss, Hendrik and Ghorai, Prasanta and Kraus, Anja and Dove, Stefan and Buschauer, Armin and Seifert, Roland (2007) Point mutations in the second extracellular loop of the histamine H-2 receptor do the species-selective activity of not affect guanidine-type agonists. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 376 (4). pp. 253-264. ISSN 0028-1298

R

Reher, T. and Brunskole, I and Burhenne, H. and Neumann, D. and Seifert, R. (2012) Differences in Histamine-H-2-Receptor-Mediated Increases in cAMP Concentration and Reactive Oxygen Species Formation in Human Eosinophils and Neutrophils. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 385 (1Suppl). S73. ISSN 0028-1298

Reinartz, Michael T. and Kaelble, Solveig and Littmann, Timo and Ozawa, Takeaki and Dove, Stefan and Kaever, Volkhard and Wainer, Irving W. and Seifert, Roland (2015) Structure-bias relationships for fenoterol stereoisomers in six molecular and cellular assays at the beta(2)-adrenoceptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 388 (1). pp. 51-65. ISSN 0028-1298, 1432-1912

Reinartz, Michael T. and Littmann, Timo and Wainer, Irving William and Ozawa, Takeaki and Dove, Stefan and Seifert, Roland (2014) Quantifying ligand bias of enantiopure fenoterol derivatives in molecular and cellular beta(2)-adrenergic assay systems. SPRINGER, NEW YORK.

S

Scharrenbroich, Jessica and Kaever, Volkhard and Dove, Stefan and Seifert, Roland and Schneider, Erich H. (2019) Hydrolysis of the non-canonical cyclic nucleotide cUMP by PDE9A: kinetics and binding mode. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 392 (2). pp. 199-208. ISSN 0028-1298, 1432-1912

Schertl, Sabine and Hartmann, Rolf W. and Batzl-Hartmann, Christine and Spruss, Thilo and Maucher, Anton and von Angerer, Erwin and Schiller, Claus D. and Schneider, Martin R. and Gust, Ronald and Schoenenberger, Helmut (2007) Platinum(II) complexes interfering with testicular steroid biosynthesis: drugs for the therapy of advanced or recurrent prostate cancers? Preclinical studies. JOURNAL OF CANCER RESEARCH AND CLINICAL ONCOLOGY, 133 (3). pp. 153-167. ISSN 0171-5216

Schneider, E. and Schreiber, E. and Bernhardt, G. and Buschauer, Armin (2005) Combined determination of binding affinity, selectivity and activity of NPY receptor ligands by multiparametric flow cytometry. In: 46th Spring Meeting of the Deutsche Gesellschaft fuer Experimentelle und Klinische Pharmakologie und Toxikologie, March 15-17, 2005, Mainz, Germany.

Schnell, David and Brunskole, Irena and Ladova, Katerina and Schneider, Erich H. and Igel, Patrick and Dove, Stefan and Buschauer, Armin and Seifert, Roland (2011) Expression and functional properties of canine, rat, and murine histamine H-4 receptors in Sf9 insect cells. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 383 (5). pp. 457-470. ISSN 0028-1298, 1432-1912

Seibel, U. and Buschauer, A. and Bernhardt, G. and Strasser, A. (2019) Dynamic mass redistribution analysis of histamine H4 receptor ligands in HEK293T cells. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 392 (1Suppl). S27-S28. ISSN 0028-1298, 1432-1912

Seifert, Roland and Xie, S. X. and Ghorai, P. and Kraus, A. and Elz, S. and Buschauer, Armin (2005) Species-selective histamine H-1-receptor activation by N-G-acylated imidazolylpropyl guanidines. In: 46th Spring Meeting of the Deutsche Gesellschaft fuer Experimentelle und Klinische Pharmakologie und Toxikologie, March 15-17, 2005, Mainz, Germany.

Strasser, Andrea and Wittmann, Hans-Joachim (2010) Distinct interactions between the human adrenergic beta(2) receptor and G alpha(s)-an in silico study. JOURNAL OF MOLECULAR MODELING, 16 (8). pp. 1307-1318. ISSN 1610-2940

Strasser, Andrea and Wittmann, Hans-Joachim (2010) In silico analysis of the histaprodifen induced activation pathway of the guinea-pig histamine H-1-receptor. JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 24 (9). pp. 759-769. ISSN 0920-654X, 1573-4951

Strasser, Andrea and Wittmann, Hans-Joachim (2007) LigPath: a module for predictive calculation of a ligand's pathway into a receptor-application to the gpH(1)-receptor. JOURNAL OF MOLECULAR MODELING, 13 (1). pp. 209-218. ISSN 1610-2940

Strasser, Andrea and Wittmann, Hans-Joachim (2013) Molecular modeling studies give hint for the existence of a symmetric h beta R-2-G alpha beta gamma-homodimer. JOURNAL OF MOLECULAR MODELING, 19 (10). pp. 4443-4457. ISSN 1610-2940, 0948-5023

Strasser, Andrea and Wittmann, Hans-Joachim and Schneider, Erich H. and Seifert, Roland (2015) Modulation of GPCRs by monovalent cations and anions. SPRINGER, NEW YORK.

T

Taha, Hesham and Dove, Stefan and Geduhn, Jens and Koenig, Burkhard and Shen, Yuequan and Tang, Wei-Jen and Seifert, Roland (2012) Inhibition of the adenylyl cyclase toxin, edema factor, from Bacillus anthracis by a series of 18 mono- and bis-(M)ANT-substituted nucleoside 5'-triphosphates. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 385 (1). pp. 57-68. ISSN 0028-1298, 1432-1912

W

Wagner, Eva and Wittmann, Hans-Joachim and Elz, Sigurd and Strasser, Andrea (2014) Pharmacological profile of astemizole-derived compounds at the histamine H-1 and H-4 receptor-H-1/H-4 receptor selectivity. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 387 (3). pp. 235-250. ISSN 0028-1298, 1432-1912

Weiss, Thomas S. and Bernhardt, Guenther and Buschauer, Armin and Thasler, Wolfgang E. and Dolgner, Doris and Zirngibl, Hubert and Jauch, Karl-Walter (2002) Polyamine levels of human colorectal adenocarcinomas are correlated with tumor stage and grade. INTERNATIONAL JOURNAL OF COLORECTAL DISEASE, 17 (6). pp. 381-387. ISSN 0179-1958, 1432-1262

Werner, Kristin and Kaelble, Solveig and Wolter, Sabine and Schneider, Erich H. and Buschauer, Armin and Neumann, Detlef and Seifert, Roland (2015) Flow cytometric analysis with a fluorescently labeled formyl peptide receptor ligand as a new method to study the pharmacological profile of the histamine H-2 receptor. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 388 (10). pp. 1039-1052. ISSN 0028-1298, 1432-1912

Wittmann, Hans-Joachim and Elz, Sigurd and Seifert, Roland and Strasser, Andrea (2011) N (alpha)-Methylated phenylhistamines exhibit affinity to the hH(4)R-a pharmacological and molecular modelling study. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 384 (3). pp. 287-299. ISSN 0028-1298, 1432-1912

Wittmann, Hans-Joachim and Seifert, Roland and Strasser, Andrea (2014) Sodium binding to hH(3)R and hH(4)R - a molecular modeling study. JOURNAL OF MOLECULAR MODELING, 20 (8): 2394. ISSN 1610-2940, 0948-5023

Wolter, Sabine and Dove, Stefan and Golombek, Marina and Schwede, Frank and Seifert, Roland (2014) N-4-monobutyryl-cCMP activates PKA RI alpha and PKA RII alpha more potently and with higher efficacy than PKG I alpha in vitro but not in vivo. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 387 (12). pp. 1163-1175. ISSN 0028-1298, 1432-1912